Histone lysine methyltransferases, like G9a, play central roles in the regulation of gene expression. A current study by Kubicek et al.  reports the identification of a G9a small-molecule inhibitor, thereby opening the way to new epigenetic cancer therapies. © 2007 Elsevier Ltd. All rights reserved.
Shaaban, S. A., & Bedford, M. T. (2007, March). Reprogramming the Histone Code. Chemistry and Biology. https://doi.org/10.1016/j.chembiol.2007.03.001