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Venkatesan Jayaprakash

  • PhD
  • Associate Professor
  • Birla Institute of Technology
  • 15h-indexImpact measure calculated using publication and citation counts. Updated daily.
  • 692CitationsNumber of citations received by Venkatesan's publications. Updated daily.

Research interests

Medicinal Chemistry; Drug Design; Molecular Modeling

About

Basically a synthetic medicinal chemist, completed PhD in Pharmacy from Birla Institute of Technology in the Title "Design, Synthesis and Pharmacological Screening of Mycobactin Analogues" Area of interest includes Molecular modeling and drug design and synthesis of small molecule heterocycles against targets of therapeutical importance. Molecular modeling includes Structure Based Drug Design (SBDD), Fragment Based Drug Design (FBDD), High-throughput Virtual Screening (HTVS) and Molecular Dynamics (MD). Targets under investigation are (i) Biosynthetic enzymes in the pathway of Mycobactin synthesis-target for anti-tubercular drug design; (ii) Histone deacetylase and Ribonucleotide-anti-cancer; (iii) protease, methyl-transferase & E-protein-anti-viral and (iv) MAO-neurodegenerative disorder. Chemical scaffolds designed: pyrazolines, aminothiazoles, thiosemicarbazones and piperazines.

Co-authors (184)

  • Soumendranath Bhakat

Publications (5)

  • Monoamine oxidase-A inhibitory activity of novel Curcumin analogues

    • Badavath V
    • Baysal İ
    • Ucar G
    • et al.
    N/AReaders
    N/ACitations
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  • Synthesis and Antiviral Activity of Dihydropyrimidines - Ciprofloxacin Mannich bases Against Various Viral Strains

    • Alavala R
    • Kulandaivelu U
    • Bonagiri P
    • et al.
    N/AReaders
    N/ACitations
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  • Chikungunya epidemiological survey and Current available inhibitors

    • Jadav S
    • Korupolu P
    • Sinha B
    • et al.
    N/AReaders
    N/ACitations
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  • X-ray crystal structure of N-benzyl-2-(4,6-diaminopyrimidin-2-ylthio)-acetamide

    • Timiri A
    • Subasri S
    • Vijayan V
    • et al.
    N/AReaders
    N/ACitations
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  • Aryl pyrazoline analogs as selective MAO-A inhibitors: further structural modification by switching the aromatic substituent

    • Basu A
    • Baysal I
    • Jagrat M
    • et al.
    N/AReaders
    N/ACitations

Editorships

Journal of Pharmaceutical Chemistry

Editor

2014 - Present

Professional experience

Associate Professor

Birla Institute of Technology

June 2016 - Present

Education

PhD

Birla Institute of Technology

January 2005 - January 2012(7 years)

PGDCAQM

University of Hyderabad

January 2003 - January 2004(a year)

M. Pharmacy

Institute of Technology Banaras Hindu University

January 1997 - January 1999(2 years)

B. Pharmacy

Madras Medical College

January 1993 - January 1996(3 years)

D. Pharmacy

Coimbatore Medical College

January 1991 - January 1992(a year)