Abstract
We report radiolabeling of thiol-containing substratesviaPd-catalyzedS-arylation with 2-[18F]fluoro-5-iodopyridine, which is readily accessible using the “minimalist” radiofluorination method. The practicality of the procedure was confirmed by preparation of a novel PSMA-specific PET-tracer as well as labeling of glutathione, Aβ oligomer-binding RD2 peptide, bovine serum albumin and PSMA I&S.
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APA
Humpert, S., Omrane, M. A., Urusova, E. A., Gremer, L., Willbold, D., Endepols, H., … Zlatopolskiy, B. D. (2021). Rapid18F-labelingviaPd-catalyzedS-arylation in aqueous medium. Chemical Communications, 57(29), 3547–3550. https://doi.org/10.1039/d1cc00745a
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