Abstract
The enantioselective formation of stereocenters proximal to unprotected heterocycles has been accomplished. Thus, vinyl boronic acids are added to heterocycle-appended enones via a modified-BINOL catalyst. Catalyst design was key to enable a general reaction. High yields and useful er's are observed for a host of common heteroaryls. © 2012 American Chemical Society.
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CITATION STYLE
APA
Le, P. Q., Nguyen, T. S., & May, J. A. (2012). A general method for the enantioselective synthesis of α-chiral heterocycles. Organic Letters, 14(23), 6104–6107. https://doi.org/10.1021/ol3030605
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